Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry, Band 31) - encadernado, livro de bolso
2006, ISBN: 9783527313686
Series Editor: Mannhold, Raimund, Series Editor: Kubinyi, Hugo, Series Editor: Folkers, Gerd, Wiley-VCH Verlag GmbH & Co. KGaA, Gebundene Ausgabe, Auflage: 2. Auflage, 207 Seiten, Publizi… mais…
amazon.de AnybookLtd Gut Custos de envio:Auf Lager. Die angegebenen Versandkosten können von den tatsächlichen Kosten abweichen. (EUR 3.00) Details... |
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry, Band 31) - encadernado, livro de bolso
2006, ISBN: 9783527313686
Series Editor: Mannhold, Raimund, Series Editor: Kubinyi, Hugo, Series Editor: Folkers, Gerd, Wiley-VCH Verlag GmbH & Co. KGaA, Gebundene Ausgabe, Auflage: 2. Auflage, 207 Seiten, Publizi… mais…
amazon.de Association Terroirs Intemporels Custos de envio:Auf Lager. Die angegebenen Versandkosten können von den tatsächlichen Kosten abweichen. (EUR 3.00) Details... |
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry) - encadernado, livro de bolso
2006, ISBN: 9783527313686
Wiley-VCH, 2006-05-02. 2. Hardcover. Used:Good., Wiley-VCH, 2006-05-02
Biblio.com |
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry) - encadernado, livro de bolso
2006, ISBN: 9783527313686
Wiley-VCH, 2006-05-02. Hardcover. Good., Wiley-VCH, 2006-05-02
Biblio.com |
2006, ISBN: 9783527313686
Wiley-VCH, 2006-05-02. Hardcover. Good., Wiley-VCH, 2006-05-02
Biblio.com |
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry, Band 31) - encadernado, livro de bolso
2006, ISBN: 9783527313686
Series Editor: Mannhold, Raimund, Series Editor: Kubinyi, Hugo, Series Editor: Folkers, Gerd, Wiley-VCH Verlag GmbH & Co. KGaA, Gebundene Ausgabe, Auflage: 2. Auflage, 207 Seiten, Publizi… mais…
Smith, Dennis A. Waterbeemd, Han van de, Walker, Don K.:
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry, Band 31) - encadernado, livro de bolso2006, ISBN: 9783527313686
Series Editor: Mannhold, Raimund, Series Editor: Kubinyi, Hugo, Series Editor: Folkers, Gerd, Wiley-VCH Verlag GmbH & Co. KGaA, Gebundene Ausgabe, Auflage: 2. Auflage, 207 Seiten, Publizi… mais…
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry) - encadernado, livro de bolso
2006
ISBN: 9783527313686
Wiley-VCH, 2006-05-02. 2. Hardcover. Used:Good., Wiley-VCH, 2006-05-02
no/na Biblio.com
Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry) - encadernado, livro de bolso
2006, ISBN: 9783527313686
Wiley-VCH, 2006-05-02. Hardcover. Good., Wiley-VCH, 2006-05-02
no/na Biblio.com
2006, ISBN: 9783527313686
Wiley-VCH, 2006-05-02. Hardcover. Good., Wiley-VCH, 2006-05-02
Dados bibliográficos do melhor livro correspondente
Autor: | |
Título: | |
Número ISBN: |
Dados detalhados do livro - Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry, Band 31)
EAN (ISBN-13): 9783527313686
ISBN (ISBN-10): 3527313680
Livro de capa dura
Ano de publicação: 2006
Editor/Editora: Wiley-VCH Verlag GmbH & Co. KGaA
187 Páginas
Peso: 0,609 kg
Língua: eng/Englisch
Livro na base de dados desde 2007-05-30T14:46:56+01:00 (Lisbon)
Página de detalhes modificada pela última vez em 2022-05-21T00:33:30+01:00 (Lisbon)
Número ISBN/EAN: 9783527313686
Número ISBN - Ortografia alternativa:
3-527-31368-0, 978-3-527-31368-6
Ortografia alternativa e termos de pesquisa relacionados:
Autor do livro: gerd folkers, raimund, hugo kubinyi, dennis smith, walker, han, van waterbeemd, don smith
Título do livro: drug metabolism, design methods, methods and principles medicinal chemistry, metabol, meta design, pharmacokinetics drugs
Dados da editora
Autor: Dennis A. Smith; Han van de Waterbeemd; Don K. Walker
Título: Methods and Principles in Medicinal Chemistry; Pharmacokinetics and Metabolism in Drug Design
Editora: Wiley-VCH
187 Páginas
Ano de publicação: 2006-02-20
Peso: 0,520 kg
Língua: Inglês
125,00 € (DE)
Not available (reason unspecified)
BB; GB; Hardcover, Softcover / Chemie; Verstehen; Pharmakokinetik; Arzneimitteldesign
PHYSICOCHEMISTRY Partition and Distribution Coefficient as Measures of Lipophilicity Limitations on the Use of Octanol Further Understanding of log P Alternative Lipophilicity Scales Computational Approaches to Lipophilicity Membrane Systems to Study Drug Behaviour NEW: Dissolution and Solubility NEW: Ionisation (pKa) PHARMACOKINETICS Intravenous Administration: Volume of Distribution Intravenous Administration: Clearance Clearance and Half-Life Intravenous administration: Infusion Oral Administration Repeated Doses Development of the Unbound (Free) Drug Model Unbound Drug and Drug Action Unbound Drug Model and Barriers to Equilibrium Slow Offset Compounds Factors Governing Unbound Drug Concentration ABSORPTION The Absorption Process Dissolution Membrane Transfer Barriers to Membrane Transfer Models for Absorption Estimation Estimation of Absorption Potential Computational Approaches DISTRIBUTION Membrane Transfer Access to the Target Brain penetration Volume of Distribution and Duration Distribution and Tmax CLEARANCE The Clearance Processes Role of Transport Proteins in Drug Clearance Interplay Between Metabolic and Renal Clearance Role of Lipophilicity in Drug Clearance RENAL CLEARANCE Kidney Anatomy and Function Lipophilicity and Reabsorption by the Kidney Effect of Charge on Renal Clearance Plasma Protein Binding and Renal Clearance Balancing Renal Clearance and Absorption Renal Clearance and Drug Design METABOLIC (HEPATIC) CLEARANCE Function of Metabolism (Biotransformation) Cytochrome P450 Other oxidative processes Oxidative Metablism and Drug Design Non-Specific Esterases Prodrugs to Aid Membrane Transfer Enzymes Catalysing Drug Conjugation Stability to Conjugation Processes Pharmacodynamics and Conjugation TOXICITY Toxicity Findings Importance of dose size Toxicity of selected compound classes Stratification of Toxicity Toxicity Prediction - Computational Toxicology Toxicogenomics Enzyme Induction (CYP3A4) and Drug Design Enzyme Inhibition and Drug Design INTERSPECIES SCALING Objectives of Allometric Scaling Allometric Scaling Species Scaling: Adjusting for Maximum Life-Span Potential Species Scaling: Incorporating Differences in Metabolic Clearance Inter-Species Scaling for Clearance by Hepatic Uptake Elimination Half-Life NEW: Scaling to pharmacological effect NEW: Single animal scaling HIGH(ER) THROUGHPUT ADME STUDIES The HTS Trend Drug Metabolism and Discovery Screening Sequences Physicochemistry Absorption / Permeability Pharmacokinetics NEW: Metabolism and Inhibition NEW: The concept of ADME space Computational Approaches in PK and Metabolism Prediction OutlookOutros livros adicionais, que poderiam ser muito similares com este livro:
Último livro semelhante:
9783527600212 Pharmacokinetics and Metabolism in Drug Design (Dennis A. Smith; Han van de Waterbeemd; Don K. Walker; Raimund Mannhold)
- 9783527600212 Pharmacokinetics and Metabolism in Drug Design (Dennis A. Smith; Han van de Waterbeemd; Don K. Walker; Raimund Mannhold)
- 9783527608225 Pharmacokinetics and Metabolism in Drug Design (Dennis A. Smith; Han van de Waterbeemd; Don K. Walker)
- 9783527329540 Pharmacokinetics and Metabolism in Drug Design (Dennis A. Smith Charlotte Allerton Amit S. Kalgutkar Han van de Waterbeemd Don K. Walker)
- 9783527301973 Pharmacokinetics and Metabolism in Drug Design (Methods and Principles in Medicinal Chemistry) (Smith, Dennis A, Waterbeemd, Han van de, Walker, Don K)
- 9783527645305 Pharmacokinetics and Metabolism in Drug Design (Dennis A. Smith; Charlotte Allerton; Amit S. Kalgutkar; Han van de Waterbeemd; Don K. Walker)
< Para arquivar...